Lamblin, M., Spingarn, R., Wang, T.T., Burger, M.C., Dabbas, B., Moitessier, N., White, J.H. and Gleason, J.L. (2010) An o-aminoaniline analogue of 1α,25-dihydroxyvitamin D3 functions as a strong vitamin D receptor antagonist. Journal of Medicinal Chemistry, 53, 7461-7465.